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  1. Pharmacological hallmarks of allostery at the M4 muscarinic receptor elucidated through structure and dynamics

    1. Ziva Vuckovic
    2. Jinan Wang
    3. Vi Pham
    4. Jesse I. Mobbs
    5. Matthew J. Belousoff
    6. Apurba Bhattarai
    7. Wessel A.C. Burger
    8. Geoff Thompson
    9. Mahmuda Yeasmin
    10. Katie Leach
    11. Emma T. van der Westhuizen
    12. Elham Khajehali
    13. Yi-Lynn Liang
    14. Alisa Glukhova
    15. Denise Wootten
    16. Craig W. Lindsley
    17. Andrew B. Tobin
    18. Patrick M. Sexton
    19. Radostin Danev
    20. Celine Valant
    21. Yinglong Miao
    22. Arthur Christopoulos
    23. David M. Thal
    This article has 5 evaluationsAppears in 2 listsLatest version Latest activity
  2. A Single Multipurpose FSH–Blocking Therapeutic for Osteoporosis and Obesity

    1. Sakshi Gera
    2. Tan-Chun Kuo
    3. Funda Korkmaz
    4. Damini Sant
    5. Victoria DeMambro
    6. Anisa Gumerova
    7. Kathayani Sudha
    8. Ashley Padilla
    9. Geoffrey Prevot
    10. Jazz Munitz
    11. Abraham Teunissen
    12. Mandy van Leent
    13. Tomas G.J.M. Post
    14. Jessica C. Fernandes
    15. Jessica Netto
    16. Farhath Sultana
    17. Eleanor Shelly
    18. Pushkar Kumar
    19. Liam Cullen
    20. Jiya Chatterjee
    21. Sari Miyashita
    22. Hasni Kannangara
    23. Megha Bhongade
    24. Kseniia Ievleva
    25. Valeriia Muradova
    26. Rogerio Batista
    27. Cemre Robinson
    28. Anne Macdonald
    29. Susan Babunovic
    30. Mansi Saxena
    31. Marcia Meseck
    32. John Caminis
    33. Jameel Iqbal
    34. Maria I. New
    35. Vitaly Ryu
    36. Se-Min Kim
    37. Jay J. Cao
    38. Neeha Zaidi
    39. Zahi Fayad
    40. Daria Lizneva
    41. Clifford J. Rosen
    42. Tony Yuen
    43. Mone Zaidi
    This article has 3 evaluationsAppears in 2 listsLatest version Latest activity
  3. Effector membrane translocation biosensors reveal G protein and βarrestin coupling profiles of 100 therapeutically relevant GPCRs

    1. Charlotte Avet
    2. Arturo Mancini
    3. Billy Breton
    4. Christian Le Gouill
    5. Alexander S. Hauser
    6. Claire Normand
    7. Hiroyuki Kobayashi
    8. Florence Gross
    9. Mireille Hogue
    10. Viktoriya Lukasheva
    11. Stéphane St-Onge
    12. Marilyn Carrier
    13. Madeleine Héroux
    14. Sandra Morissette
    15. Eric Fauman
    16. Jean-Philippe Fortin
    17. Stephan Schann
    18. Xavier Leroy
    19. David E. Gloriam
    20. Michel Bouvier
    This article has 4 evaluationsAppears in 2 listsLatest version Latest activity
  4. Common coupling map advances GPCR-G protein selectivity

    1. Alexander S. Hauser
    2. Charlotte Avet
    3. Claire Normand
    4. Arturo Mancini
    5. Asuka Inoue
    6. Michel Bouvier
    7. David E. Gloriam
    This article has 4 evaluationsAppears in 2 listsLatest version Latest activity
  5. NBI-921352, a First-in-Class, Na V 1.6 Selective, Sodium Channel Inhibitor That Prevents Seizures in Scn8a Gain-of-Function Mice, and Wild-Type Mice and Rats

    1. JP Johnson
    2. Thilo Focken
    3. Kuldip Khakh
    4. Parisa Karimi Tari
    5. Celine Dube
    6. Aaron Williams
    7. Jean-Christophe Andrez
    8. Girish Bankar
    9. David Bogucki
    10. Kristen Burford
    11. Elaine Chang
    12. Sultan Chowdhury
    13. Richard Dean
    14. Gina de Boer
    15. Shannon Decker
    16. Christoph Dehnhardt
    17. Mandy Feng
    18. Wei Gong
    19. Samuel J Goodchild
    20. Michael Grimwood
    21. Abid Hasan
    22. Angela Hussainkhel
    23. Qi Jia
    24. Stephanie Lee
    25. Jenny Li
    26. Sophia Lin
    27. Andrea Lindgren
    28. Verner Lofstrand
    29. Janette Mezeyova
    30. Rostam Namdari
    31. Karen Nelkenbrecher
    32. Noah Gregory Shuart
    33. Luis Sojo
    34. Shaoyi Sun
    35. Matthew Taron
    36. Matthew Waldbrook
    37. Diana Weeratunge
    38. Steven Wesolowski
    39. Michael Wilson
    40. Zhiwei Xie
    41. Rhena Yoo
    42. Clint Young
    43. Alla Zenova
    44. Wei Zhang
    45. Alison J Cutts
    46. Robin P Sherrington
    47. Simon N Pimstone
    48. Raymond Winquist
    49. Charles J Cohen
    50. James R Empfield
    This article has 4 evaluationsAppears in 2 listsLatest version Latest activity
  6. Fluorescence Activation Mechanism and Imaging of Drug Permeation with New Sensors for Smoking-Cessation Ligands

    1. Aaron L. Nichols
    2. Zack Blumenfeld
    3. Chengcheng Fan
    4. Laura Luebbert
    5. Annet E. M. Blom
    6. Bruce N. Cohen
    7. Jonathan S. Marvin
    8. Philip M. Borden
    9. Charlene H. Kim
    10. Anand K. Muthusamy
    11. Amol V. Shivange
    12. Hailey J. Knox
    13. Hugo Rego Campello
    14. Jonathan H. Wang
    15. Dennis A. Dougherty
    16. Loren L. Looger
    17. Timothy Gallagher
    18. Douglas C. Rees
    19. Henry A. Lester
    This article has 4 evaluationsAppears in 2 listsLatest version Latest activity